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Properties of substance:

[Dmt1, (R)-βPro2, (2-Furyl)Map4]endomorphin-1



skc-file

Group of substances:

organic

Empirical formula (Hill's system for organic substances):

C35H40N6O6

Molar/atomic mass: 640.729

Melting point (°C):

150-153

Numerical data:

μ-Opioid Receptor Binding (nM): 0.00372
κ-Opioid Receptor Binding (nM): 205
δ-Opioid Receptor Binding (nM): 19.8

References:

  1. Liu X., Wang Y., Xing Y., Yu J., Ji H., Kai M., Wang Z., Wang D., Zhang Y., Zhao D., Wang R. Design, Synthesis, and Pharmacological Characterization of Novel Endomorphin-1 Analogues as Extremely Potent μ-Opioid Agonists / Journal of Medicinal Chemistry. - 2013. - Vol. 56, No. 7. - pp. 3102-3114

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    © Collected Ruslan Anatolievich Kiper, burewestnik@mail.ru